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Felypressin
drug data and news
Felypressin drug data, resources, and news articles (when available). Onconews.org provides news on cancer research. This section, which includes profiles on medicines that may or not be cancer-related is in beta form. If things run smoothly we will be releasing a new format late in the summer of 2006.
| Generic name |
Felypressin
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| Brand Names/Synonyms |
FELYPRESSIN; 2-(L-Phenylalanine)-8-L-lysinevasopressin; FELYPRESSIN; Felipressina [DCIT]; Felipresina [INN-Spanish]; Felypressine [INN-French]; Felypressinum [INN-Latin]; Felypressin [USAN:BAN:INN] |
| Indication |
Local anaesthetic |
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Description |
Synthetic analog of LYPRESSIN with more vasoconstrictor than antidiuretic action. It is used as a hemostatic |
| Pharmacology |
Used as a localizing agent for anesthetics. Felypressin is a synthetic analog of lypressin or vasopressin with more vasoconstrictor activity than antidiuretic action. It is used primarily as a hemostatic. |
| Mechanism Of Action |
Binds to the vasopressin receptor V1a. This causes contraction of the smooth muscle in the vascular bed, especially capillaries, small arterioles and venules. |
Felypressin News
(When available) |
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| Dosage Forms |
Not Available |
| Drug_Category |
Vasoconstrictor Agents; Renal Agents; Hemostatics (20:12.16); |
| Absorption |
Not Available |
| Interactions |
Not Available |
| Toxicity |
Not Available |
| Organisms Affected |
Humans and other mammals |
| Chemical IUPAC Name |
N-[5-amino-1-(carbamoylmethylcarbamoyl)pentyl]-1-[[19-amino-13,16-dibenzyl-10-(2-carbamoylethyl)-7-(carbamoylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicos-4-yl]carbonyl]pyrrolidine-2-carboxamide |
| Chemical Formula |
C46H65N13O11S2 |
| Molecular Weight |
1040.22 g/mol |
| Smiles String |
C1CC(N(C1)C(=O)C2CSSCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=CC=C4)N)C(=O)NC(CCCCN)C(=O)NCC(=O)N |
| Melting Point |
Not Available |
| Water Solubility |
Not Available |
| State |
Solid |
| LogP/Hphobicity |
-3.351 |
| Isoelectric Point |
Not Available |
| Biotransformation |
Not Available |
| Half Life |
Not Available |
| Protein Binding [%] |
Not Available |
| RxList Link |
Not Available>RXlist |
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| Drug Reference |
Not Available |
| Drug Type |
Approved Drug |
| Accession No |
BIOD00114 |
| CAS Registry Number |
56-59-7 |
| KEGG Compound ID |
Not Available |
| PubChem ID |
SID:148784 |
| PharmGKB ID |
Not Available |
| SwissProt ID |
Not Available |
| GenBank ID |
Not Available |
| Drug ID Number [DIN] |
Not Available
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